Program

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Lectures

Sunday, Aug 25, 2024

16.00
Welcome and Summer School Opening
16.30

Prof. Dirk Trauner, University of Pennsylvania (US)
«On the Clinical Relevance of Photopharmacology»

18.30
Dinner
20.00

Get together

Monday, Aug 26, 2024

08.30

tba,
«open»

09.30

Prof. Stefan Arold, King Abdullah University of Science and Technology, KAUST (SA)
«Chemical Competition by Biological Design: Function from Noise?»

10.30
Coffee Break
11.00

Prof. Anna Mapp, University of Michigan (USA)
«Strategies for Drugging Transcription Factors: Lessons from Nature Privileged Scaffolds for Modulating Dynamic Protein-Protein Interactions»

12.00

Dr. Guido Koch, Amphilix, SynpleChem, eMolecules (CH)
«Medicinal Chemistry of Kinase Drug Discovery – Case Studies and Future Directions»

13.00
Lunch Break

14.30

Workshop in Teams

16.00

Coffee Break

16.30

Short Communications Session A

18.30
Dinner
20.00
Poster Session A

Tuesday, Aug 27, 2024

08.30

Prof. Brian Paegel, University of California, Irvine (USA)
«Scaling Probe Discovery to the Proteome via Selective Translation Modulation»

09.30

Prof. Ben Schumann, Imperial College London (UK)
«Bump-and-hole Engineering of Glycosyltransferases to Dissect Protein Glycosylation»

10.30
Coffee Break
11.00

tba,
«open»

12.00

Industry Lecture
Ahmed Mahmoud, Chemspeed
Translating your Processes to Automation for Accelerated Research and Development


13.00

Lunch Break & Excursion

18.30
Dinner
20.00
Poster Session B

Wednesday, Aug 28, 2024

08.30

Prof. Stefan Arold, King Abdullah University of Science and Technology, KAUST (SA)
«The Good, the Bad, and the Fortuitous: Chemical Blobology in Structural Biology»

09.30

Prof. Brian PaegelUniversity of California, Irvine (USA)
«Scaling Pharmacokinetic Analysis to Chart Chemical Space Beyond the Rule-of-5»

10.30
Coffee Break
11.00

Prof. Anna Mapp, University of Michigan (USA)
«Strategies for Drugging Transcription Factors: Lessons from Nature Privileged Scaffolds for Modulating Dynamic Protein-Protein Interactions»

12.00

Dr. Jingwen Shi & Dr. Sacha Javor, Space Pharmaceuticals AG
«tba.»

13.00
Lunch Break

14.30

Workshop in Teams

16.00

Coffee Break

16.30

Short Communications Session B

18.30

Conference Dinner & Awards

Thursday, Aug 29, 2024

08.30

Prof. Ben Schumann, Imperial College London (UK)
«Cell-specific Bioorthogonal Tagging of Glycoproteins»

09.30

Prof. Dirk Trauner, University of Pennsylvania (USA)
«On the Clinical Relevance of Total Synthesis»

10.30
Coffee Break
11.00

Closure